Acyclovir molecular structure

Acyclovir

Also known as: Zovirax, Acivir, Herpex, Cyclovir, Ocuvir

CAS Number: 59277-89-3

Antiviral (Nucleoside Analogue, Anti-Herpes)

Pharmacopeia Standards

USPIPEPBPJPWHO

Mechanism of Action

Acyclovir is an acyclic guanosine analogue that is selectively monophosphorylated by herpesvirus-encoded thymidine kinase, so activation is largely confined to infected cells. Host guanylate kinase and other cellular kinases complete conversion to acyclovir triphosphate, which competitively inhibits viral DNA polymerase far more potently than the host enzyme. Incorporation into the elongating DNA strand causes obligate chain termination and inactivates the polymerase.

Technical Specifications

Generic / INN NameAcyclovir
CAS Registry Number59277-89-3
Molecular FormulaC8H11N5O3
Molecular Weight225.20 g/mol g/mol
Typical PurityNot less than 98.0% and not more than 101.0% on anhydrous basis (USP/EP)
Storage ConditionsStore below 30 degrees C in well-closed containers protected from light and moisture.
Shelf Life60 months from date of manufacture in original sealed packing
CategoryAntivirals

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Bulk API for oral tablets, dispersible tablets and suspensions, topical creams and ointments, ophthalmic ointments, and sterile acyclovir sodium powder for intravenous infusion.

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