Amphotericin B molecular structure

Amphotericin B

Also known as: Fungizone, AmBisome, Abelcet, Amphotec, Fungisome, Amphonex

CAS Number: 1397-89-3

Polyene macrolide antifungal — systemic, broad spectrum

Pharmacopeia Standards

USPBPEPIPJPCP

Mechanism of Action

Amphotericin B binds ergosterol in the fungal membrane and forms ion-permeable channels, and also extracts ergosterol directly out of the bilayer into extramembranous aggregates. Both mechanisms collapse the transmembrane electrochemical gradient and cause rapid fungicidal killing. Residual affinity for mammalian cholesterol underlies its nephrotoxicity, which is what drove development of the liposomal and lipid-complex presentations.

Technical Specifications

Generic / INN NameAmphotericin B
CAS Registry Number1397-89-3
Molecular FormulaC47H73NO17
Molecular Weight924.08 g/mol
Typical PurityNot less than 750 µg/mg (on dried basis); amphotericin A not more than 5.0%
Storage ConditionsStore at 2–8°C in tightly closed, light-resistant containers under nitrogen; protect from light, heat and moisture
Shelf Life36 months from date of manufacture when stored refrigerated
CategoryAntifungals

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Invasive candidiasis and candidaemia, cryptococcal meningitis, invasive aspergillosis, mucormycosis, visceral leishmaniasis, disseminated histoplasmosis, blastomycosis and coccidioidomycosis

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