Aztreonam molecular structure

Aztreonam

Also known as: Azactam, Cayston, Primbactam, Azenam

CAS Number: 78110-38-0

Monobactam Antibiotic (Beta-Lactam)

Pharmacopeia Standards

USPBPEPIPJP

Mechanism of Action

Aztreonam is a monocyclic beta-lactam that binds penicillin-binding protein 3 in aerobic Gram-negative bacilli with very high affinity, blocking septal peptidoglycan synthesis and causing filamentation and lysis. Its monobactam nucleus is stable to metallo-beta-lactamases, which hydrolyse virtually all other beta-lactams. It has no meaningful activity against Gram-positive organisms or anaerobes, and its structural dissimilarity to penicillins means it is generally tolerated by penicillin-allergic patients.

Technical Specifications

Generic / INN NameAztreonam
CAS Registry Number78110-38-0
Molecular FormulaC13H17N5O8S2
Molecular Weight435.43 g/mol g/mol
Typical PurityNLT 96.0% and NMT 102.0% on the anhydrous basis; endotoxin NMT 0.17 IU/mg; open-ring and isomeric impurities individually NMT 0.5%
Storage ConditionsStore below 25 C in tight, light-resistant containers under nitrogen; protect from moisture and elevated temperature.
Shelf Life36 months for sterile grade in original sealed packaging
CategoryMonobactams

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Sterile powder for injection in 500 mg, 1 g and 2 g vials; lyophilised inhalation solution for cystic fibrosis; investigational aztreonam-avibactam combinations for metallo-beta-lactamase producers.

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