Capreomycin Sulfate molecular structure

Capreomycin Sulfate

Also known as: Capastat, Capocin, Caprihans, Capreomycin Sulphate

CAS Number: 1405-37-4

Antitubercular (Cyclic Polypeptide Injectable, Second-Line)

Pharmacopeia Standards

USPBPEPWHO

Mechanism of Action

Capreomycin is a cyclic polypeptide complex of capreomycins IA and IB that binds the bacterial ribosome at the interface between the 30S and 50S subunits. It blocks the tRNA translocation step of protein synthesis in a manner mechanistically related to the aminoglycosides but through a distinct binding site. This allows activity against some strains resistant to streptomycin, though cross-resistance with kanamycin and amikacin is common through rrs and tlyA mutations.

Technical Specifications

Generic / INN NameCapreomycin Sulfate
CAS Registry Number1405-37-4
Molecular FormulaC25H44N14O8 · xH2SO4
Molecular Weight668.71 g/mol (free base); approximately 1320 g/mol as sulfate complex g/mol
Typical PurityNot less than 700 mcg of capreomycin per mg (on anhydrous basis, USP potency)
Storage ConditionsStore at 2-8 degrees C in tightly closed, moisture-proof containers; hygroscopic, protect from light and humidity
Shelf Life24 months from date of manufacture when stored refrigerated as directed
CategoryAnti-Tubercular Agents

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Bulk sterile API for 1 g capreomycin sulfate injection vials used in longer regimens for multidrug-resistant and extensively drug-resistant tuberculosis where all-oral options are unavailable.

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