Dapsone molecular structure

Dapsone

Also known as: Aczone, Avlosulfon, Dapsone DS, Diaminodiphenyl Sulfone, DDS

CAS Number: 80-08-0

Antileprotic / Sulfone Antibacterial

Pharmacopeia Standards

USPBPIPEPJPWHO

Mechanism of Action

Dapsone is a sulfone analogue of para-aminobenzoic acid that competitively inhibits dihydropteroate synthase in the bacterial folate biosynthesis pathway. Blocking dihydrofolate formation starves the organism of the tetrahydrofolate needed for purine and thymidine synthesis, giving bacteriostatic activity against Mycobacterium leprae. It also exerts a separate anti-inflammatory effect by suppressing neutrophil myeloperoxidase and chemotaxis, which underpins its dermatological uses.

Technical Specifications

Generic / INN NameDapsone
CAS Registry Number80-08-0
Molecular FormulaC12H12N2O2S
Molecular Weight248.30 g/mol g/mol
Typical Purity99.0% - 101.0% (on dried basis, USP/BP assay)
Storage ConditionsStore in tightly closed, light-resistant containers below 25 degrees C; protect from light and air to prevent discolouration
Shelf Life60 months from date of manufacture when stored as directed
CategoryAntileprotics

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Bulk API for 25 mg, 50 mg and 100 mg dapsone tablets used in WHO multidrug therapy blister packs for paucibacillary and multibacillary leprosy, plus topical 5% and 7.5% gels for acne and oral use in dermatitis herpetiformis and PCP prophylaxis.

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