Diethylcarbamazine Citrate molecular structure

Diethylcarbamazine Citrate

Also known as: Hetrazan, Banocide, Notezine, DEC, Filaria Tablets, Carbamazine

CAS Number: 1642-54-2

Antifilarial Anthelmintic (Piperazine Derivative)

Pharmacopeia Standards

USPBPIPEPWHO

Mechanism of Action

Diethylcarbamazine acts principally on the host arachidonic acid pathway, inhibiting cyclooxygenase and lipoxygenase-derived mediators so that microfilariae lose their protective surface and are rapidly sequestered and destroyed by the host innate immune system. It also appears to sensitise the parasite surface to granulocyte adherence. Its action is therefore substantially immune-dependent rather than directly cytotoxic, which explains its rapid microfilaricidal effect in the bloodstream.

Technical Specifications

Generic / INN NameDiethylcarbamazine Citrate
CAS Registry Number1642-54-2
Molecular FormulaC10H21N3O · C6H8O7
Molecular Weight391.42 g/mol g/mol
Typical PurityNot less than 98.0% (assay), on the dried basis
Storage ConditionsStore in tight, moisture-proof containers below 30°C; protect rigorously from humidity due to deliquescence
Shelf Life36–48 months in original moisture-barrier packaging
CategoryAnthelmintics

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Tablets for lymphatic filariasis mass drug administration, tropical pulmonary eosinophilia and loiasis; DEC-fortified salt programmes; triple-drug IDA regimens with ivermectin and albendazole.

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