Imipenem molecular structure

Imipenem

Also known as: Primaxin (with cilastatin), Tienam, Zienam

CAS Number: 74431-23-5

Carbapenem — broad-spectrum parenteral beta-lactam

Pharmacopeia Standards

USPEP

Mechanism of Action

First carbapenem introduced clinically; highest in vitro PBP-binding affinity. Requires co-administration with cilastatin (renal dehydropeptidase-I inhibitor) to prevent renal inactivation and nephrotoxicity. Cilastatin does not alter antibacterial activity. Active against most aerobic gram-positive, gram-negative, and anaerobic organisms.

Technical Specifications

Generic / INN NameImipenem
CAS Registry Number74431-23-5
Molecular FormulaC12H17N3O4S
Molecular Weight299.35 g/mol
Typical Purity97.0–102.0%
Storage ConditionsStore below 25°C, protected from moisture and light
Shelf Life24 months from date of manufacture
CategoryCarbapenems

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Serious polymicrobial infections requiring broad-spectrum coverage (intra-abdominal, pelvic, respiratory), complicated UTIs, bacteremia, hospital-acquired pneumonia, infections in immunocompromised patients. Used as imipenem-cilastatin combination exclusively for parenteral administration.

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