Josamycin molecular structure

Josamycin

Also known as: Josacine, Wilprafen, Josamy, Iosalide

CAS Number: 16846-24-5

Macrolide Antibacterial

Pharmacopeia Standards

JPEPCP

Mechanism of Action

Josamycin is a 16-membered macrolide that binds the 50S ribosomal subunit and blocks the peptidyl transferase centre, halting nascent chain elongation. Its 16-membered ring means it is not inactivated by the inducible erm-mediated MLSb resistance seen with 14-membered macrolides in some staphylococcal strains. Activity is bacteriostatic against Gram-positive cocci, Mycoplasma and Chlamydia.

Technical Specifications

Generic / INN NameJosamycin
CAS Registry Number16846-24-5
Molecular FormulaC42H69NO15
Molecular Weight827.99 g/mol g/mol
Typical PurityNLT 900 micrograms of josamycin per mg on the dried basis; related substances per EP/JP limits
Storage ConditionsStore below 25 degrees C in tightly closed containers, protected from light and moisture
Shelf Life36 months from date of manufacture
CategoryMacrolides

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oral tablets, dispersible tablets and dry suspensions, principally for European, Japanese, Russian and CIS markets where the molecule retains a strong prescribing base.

Manufacturers (0+)

View all →
No manufacturers listed yet. Register your company to appear here.