Nifuroxazide molecular structure

Nifuroxazide

Also known as: Ercefuryl, Antinal, Diafuryl, Pentofuryl, Enterofuryl

CAS Number: 965-52-6

Non-absorbed intestinal nitrofuran antiseptic

Pharmacopeia Standards

EP

Mechanism of Action

Nifuroxazide is reduced by enteric bacterial nitroreductases to reactive species that inhibit dehydrogenase enzymes and disrupt bacterial protein and nucleic acid synthesis. Because the molecule is essentially not absorbed from the gastrointestinal tract, activity is confined to the gut lumen and systemic exposure is negligible. It has also attracted research interest as a STAT3 signalling inhibitor, though that is not a registered use.

Technical Specifications

Generic / INN NameNifuroxazide
CAS Registry Number965-52-6
Molecular FormulaC12H9N3O5
Molecular Weight275.22 g/mol g/mol
Typical Purity98.5-101.5% on dried basis (EP); total impurities NMT 1.0%
Storage ConditionsStore in well-closed containers protected from light at 15-25 C in a dry place
Shelf Life48 months from date of manufacture
CategoryNitrofurans

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oral capsules, tablets and paediatric suspensions for acute infectious diarrhoea, marketed heavily across France, Eastern Europe, Turkey, the Middle East, North Africa and Southeast Asia.

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