Nystatin molecular structure

Nystatin

Also known as: Mycostatin, Nystan, Nystatin Oral Suspension, Candistat, Mycolog

CAS Number: 1400-61-9

Polyene macrolide antifungal — topical and oral non-absorbed

Pharmacopeia Standards

USPBPEPIPJPCP

Mechanism of Action

Nystatin binds ergosterol in the fungal plasma membrane and self-assembles into transmembrane pores, allowing uncontrolled efflux of potassium and small metabolites and causing osmotic lysis. Because the target is a sterol rather than an enzyme, acquired resistance is uncommon. Its negligible absorption from the gastrointestinal tract confines activity to the gut lumen and mucosal surfaces, which is the basis for its oral use against candidiasis without systemic toxicity.

Technical Specifications

Generic / INN NameNystatin
CAS Registry Number1400-61-9
Molecular FormulaC47H75NO17
Molecular Weight926.09 g/mol
Typical PurityNot less than 4400 IU/mg (on dried basis)
Storage ConditionsStore at 2–8°C in tightly closed, light-resistant containers under nitrogen; protect from light, heat and moisture
Shelf Life36 months from date of manufacture when stored refrigerated
CategoryAntifungals

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oropharyngeal candidiasis, oesophageal and intestinal candidiasis, cutaneous and mucocutaneous candidiasis, vulvovaginal candidiasis, prophylaxis of candidal overgrowth in neonates and immunocompromised patients

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