Ornidazole molecular structure

Ornidazole

Also known as: Tiberal, Ornidal, Ornof, Dazolic, Giro

CAS Number: 16773-42-5

Nitroimidazole antiprotozoal and antianaerobic

Pharmacopeia Standards

IPEPCP

Mechanism of Action

Ornidazole enters anaerobic organisms by passive diffusion and undergoes reduction of its 5-nitro group by low-redox-potential ferredoxin systems, generating short-lived nitro radical anions. These species cause strand breaks and helix destabilisation in microbial DNA and disable repair, killing the organism. The chlorohydroxypropyl side chain gives a longer elimination half-life than metronidazole, supporting twice-daily dosing regimens.

Technical Specifications

Generic / INN NameOrnidazole
CAS Registry Number16773-42-5
Molecular FormulaC7H10ClN3O3
Molecular Weight219.63 g/mol g/mol
Typical Purity99.0-101.0% on anhydrous basis; residual epichlorohydrin NMT 1 ppm
Storage ConditionsStore in tightly closed light-resistant containers below 25 C in a dry place
Shelf Life48 months from date of manufacture
CategoryNitroimidazoles

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oral tablets and IV infusion for amoebiasis, giardiasis, trichomoniasis and anaerobic surgical prophylaxis; widely formulated as fixed-dose combinations with ofloxacin, ciprofloxacin, levofloxacin and satranidazole.

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