Secnidazole molecular structure

Secnidazole

Also known as: Solosec, Flagentyl, Secnil, Secnidal, Sindose

CAS Number: 3366-95-8

Long-acting nitroimidazole antiprotozoal

Pharmacopeia Standards

IPEP

Mechanism of Action

Secnidazole is reduced intracellularly by anaerobic and microaerophilic organisms to nitro radical anions that damage DNA and inhibit nucleic acid synthesis, in common with the rest of the nitroimidazole class. Its distinguishing feature is a plasma half-life of roughly seventeen to twenty-nine hours, several times longer than metronidazole, which allows a complete course to be delivered as a single dose. That pharmacokinetic profile is the entire commercial rationale for the molecule.

Technical Specifications

Generic / INN NameSecnidazole
CAS Registry Number3366-95-8
Molecular FormulaC7H11N3O3
Molecular Weight185.18 g/mol g/mol
Typical Purity98.0-102.0% on anhydrous basis; total impurities NMT 1.0%
Storage ConditionsStore in well-closed containers at 15-25 C, protected from light and moisture
Shelf Life48 months from date of manufacture
CategoryNitroimidazoles

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Single-dose oral granules and tablets for bacterial vaginosis and trichomoniasis, and single-dose or short-course therapy for amoebiasis and giardiasis in emerging markets.

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