Sparfloxacin molecular structure

Sparfloxacin

Also known as: Zagam, Spara, Sparcin, Torospar

CAS Number: 110871-86-8

Fluoroquinolone Antibacterial

Pharmacopeia Standards

IPJPCP

Mechanism of Action

Sparfloxacin inhibits DNA gyrase and topoisomerase IV with enhanced Gram-positive potency conferred by the 5-amino and 8-fluoro substitutions. The dimethylpiperazinyl group at C7 extends the post-antibiotic effect and half-life. Killing is concentration dependent and bactericidal.

Technical Specifications

Generic / INN NameSparfloxacin
CAS Registry Number110871-86-8
Molecular FormulaC19H22F2N4O3
Molecular Weight392.40 g/mol g/mol
Typical PurityNLT 98.5% on the anhydrous basis; trans-isomer and des-fluoro impurities individually NMT 0.5%
Storage ConditionsStore below 25 degrees C in tightly closed light-resistant containers; protect from direct sunlight
Shelf Life48 months from date of manufacture
CategoryFluoroquinolones

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oral tablets and ophthalmic solutions, retained mainly in Indian, Japanese and Chinese markets. The 8-fluoro substitution carries a well-known phototoxicity liability that shaped its regulatory trajectory.

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