Spiramycin molecular structure

Spiramycin

Also known as: Rovamycine, Provamycin, Rovamycin, Spiramyl

CAS Number: 8025-81-8

Macrolide Antibacterial / Antiprotozoal

Pharmacopeia Standards

EPBPCPWHO

Mechanism of Action

Spiramycin binds the 50S ribosomal subunit at the peptidyl transferase region and inhibits translocation during bacterial protein synthesis. Its unusually high and persistent intracellular tissue concentrations, particularly in placental and salivary tissue, distinguish it from other 16-membered macrolides. It also suppresses Toxoplasma gondii replication, which underpins its obstetric use.

Technical Specifications

Generic / INN NameSpiramycin
CAS Registry Number8025-81-8
Molecular FormulaC43H74N2O14 (spiramycin I)
Molecular Weight843.05 g/mol (spiramycin I) g/mol
Typical PurityNLT 4100 IU/mg; spiramycin I NLT 80.0%, sum of spiramycins I, II and III NLT 90.0% (EP)
Storage ConditionsStore in airtight containers protected from light at 2-8 degrees C or below 25 degrees C per supplier specification
Shelf Life36 months from date of manufacture
CategoryMacrolides

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oral tablets and granules expressed in international units, spiramycin-metronidazole fixed-dose dental combinations, and veterinary premixes. Also supplied as spiramycin adipate and embonate salts for animal health formulators.

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