Sulfadiazine molecular structure

Sulfadiazine

Also known as: Sulfadiazine, Flamazine and Silvadene (as silver sulfadiazine), Coptin

CAS Number: 68-35-9

Sulfonamide antibacterial and antiprotozoal

Pharmacopeia Standards

USPBPIPEPJPCP

Mechanism of Action

Sulfadiazine competitively inhibits dihydropteroate synthase and blocks incorporation of para-aminobenzoic acid into dihydropteroic acid, starving susceptible bacteria and protozoa of folate. Combined with pyrimethamine it gives sequential folate blockade that is the standard regimen for toxoplasmic encephalitis. As the silver salt it additionally delivers ionic silver that denatures microbial proteins at the burn wound surface.

Technical Specifications

Generic / INN NameSulfadiazine
CAS Registry Number68-35-9
Molecular FormulaC10H10N4O2S
Molecular Weight250.28 g/mol g/mol
Typical Purity99.0-101.0% on dried basis; residue on ignition NMT 0.1%
Storage ConditionsStore in tight, light-resistant containers at 15-30 C in a dry area
Shelf Life60 months from date of manufacture
CategorySulfonamides

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oral tablets for toxoplasmosis with pyrimethamine and for rheumatic fever prophylaxis, silver sulfadiazine cream for burn wound care, and veterinary sulfonamide preparations for poultry coccidiosis.

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