Sulfadoxine molecular structure

Sulfadoxine

Also known as: Fansidar (with pyrimethamine), Sulfadar, Malostat, Amalar

CAS Number: 2447-57-6

Antimalarial / Long-Acting Sulfonamide (Antifolate)

Pharmacopeia Standards

BPIPEPWHO

Mechanism of Action

Sulfadoxine is a structural analogue of para-aminobenzoic acid that competitively inhibits parasite dihydropteroate synthase, blocking folate biosynthesis at an early step. Because malaria parasites must synthesise folate de novo rather than salvage it, this starves them of the cofactors needed for DNA synthesis. Paired with pyrimethamine, which inhibits the downstream dihydrofolate reductase, the sequential blockade is markedly synergistic.

Technical Specifications

Generic / INN NameSulfadoxine
CAS Registry Number2447-57-6
Molecular FormulaC12H14N4O4S
Molecular Weight310.33 g/mol g/mol
Typical PurityNot less than 99.0% (assay), on the dried basis
Storage ConditionsStore in well-closed, light-resistant containers below 30°C
Shelf Life60 months in original sealed packaging
CategoryAntimalarials

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Fixed-dose sulfadoxine-pyrimethamine tablets for intermittent preventive treatment in pregnancy and for seasonal malaria chemoprevention; veterinary coccidiostat formulations.

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