Tazobactam Sodium molecular structure

Tazobactam Sodium

Also known as: Zosyn (with piperacillin), Tazocin, Zerbaxa (with ceftolozane), Piptaz

CAS Number: 89785-84-2

Beta-Lactamase Inhibitor (Triazolylmethyl Penicillanic Acid Sulfone)

Pharmacopeia Standards

USPEPIPCP

Mechanism of Action

Tazobactam is a triazolylmethyl penicillanic acid sulfone that irreversibly acylates the active-site serine of class A beta-lactamases, including many extended-spectrum enzymes. The resulting stable acyl-enzyme complex prevents hydrolysis of the partner beta-lactam. Its inhibitory spectrum is broader than sulbactam and it has essentially no intrinsic antibacterial activity of its own.

Technical Specifications

Generic / INN NameTazobactam Sodium
CAS Registry Number89785-84-2
Molecular FormulaC10H11N4NaO5S
Molecular Weight322.27 g/mol g/mol
Typical PurityNLT 96.0% and NMT 102.0% on the anhydrous basis; endotoxin NMT 0.17 IU/mg for sterile grade
Storage ConditionsStore below 25 C in tight, light-resistant containers under nitrogen; hygroscopic, protect from moisture and heat.
Shelf Life24 months for sterile grade in original sealed packaging
CategoryBeta-Lactamase Inhibitors

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Piperacillin-tazobactam injection at the fixed 8:1 ratio in 2.25 g, 3.375 g and 4.5 g vials; ceftolozane-tazobactam at 2:1; cefepime-tazobactam and ceftriaxone-tazobactam combinations marketed in India.

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