Thiamphenicol molecular structure

Thiamphenicol

Also known as: Urfamycine, Thiophenicol, Glitisol, Fluimucil Antibiotic (as thiamphenicol glycinate)

CAS Number: 15318-45-3

Amphenicol antibiotic (methylsulfonyl analogue)

Pharmacopeia Standards

JPCPBP

Mechanism of Action

Thiamphenicol is the methylsulfonyl analogue of chloramphenicol and inhibits bacterial protein synthesis by binding the 50S ribosomal subunit and blocking peptidyl transferase activity. Replacing the nitro group with a methylsulfonyl group removes the nitroreduction pathway implicated in idiosyncratic aplastic anaemia, giving a markedly cleaner haematological profile. It is excreted largely unchanged in urine, which underpins its use in urogenital and respiratory indications.

Technical Specifications

Generic / INN NameThiamphenicol
CAS Registry Number15318-45-3
Molecular FormulaC12H15Cl2NO5S
Molecular Weight356.22 g/mol g/mol
Typical Purity98.0-102.0% on anhydrous basis; total impurities NMT 1.0%
Storage ConditionsStore below 25 C in tightly closed, light-resistant containers away from moisture
Shelf Life48 months from date of manufacture in original unopened packing
CategoryAmphenicols

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oral capsules and granules for respiratory and urogenital infection, thiamphenicol glycinate acetylcysteinate for inhalation and injection, and veterinary preparations for swine and poultry in markets that permit amphenicol use.

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