Tilmicosin Phosphate molecular structure

Tilmicosin Phosphate

Also known as: Micotil, Pulmotil, Pulmotil AC, Tilmovet, Tilmicin

CAS Number: 137330-13-3

Veterinary macrolide antibiotic

Pharmacopeia Standards

USPEPCP

Mechanism of Action

Tilmicosin is a semisynthetic macrolide derived from tylosin that binds the 50S ribosomal subunit and inhibits peptide chain elongation, with particular potency against Mannheimia haemolytica, Pasteurella multocida and Mycoplasma species. It accumulates to very high concentrations in lung tissue and alveolar macrophages, which sustains a therapeutic effect for several days after a single dose. That same tissue affinity makes the injectable form cardiotoxic to humans, horses and swine on accidental exposure.

Technical Specifications

Generic / INN NameTilmicosin Phosphate
CAS Registry Number137330-13-3
Molecular FormulaC46H80N2O13 . H3PO4
Molecular Weight967.13 g/mol (as the phosphate salt) g/mol
Typical PurityNLT 900 mcg tilmicosin per mg on anhydrous basis (USP); related substances within monograph limits
Storage ConditionsStore below 25 C in tightly closed containers, protect from light and moisture
Shelf Life24-36 months from date of manufacture
CategoryVeterinary Antibiotics

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Subcutaneous injection for bovine and ovine respiratory disease, oral premix and water-soluble presentations for swine and poultry respiratory disease and mycoplasmosis, and metaphylactic use in feedlot cattle.

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