Tinidazole molecular structure

Tinidazole

Also known as: Tindamax, Fasigyn, Tiniba, Trigyn, Simplotan

CAS Number: 19387-91-8

Second-generation nitroimidazole antiprotozoal and antianaerobic

Pharmacopeia Standards

USPBPIPEPCP

Mechanism of Action

Tinidazole diffuses into anaerobic bacteria and protozoa where the 5-nitro group is reduced by ferredoxin-type electron transport proteins to cytotoxic nitro radical anions. These radicals fragment DNA and inhibit further nucleic acid synthesis, producing rapid cell death. Aerobic organisms lack the low-redox-potential reduction systems required, which confines activity to anaerobes and microaerophiles.

Technical Specifications

Generic / INN NameTinidazole
CAS Registry Number19387-91-8
Molecular FormulaC8H13N3O4S
Molecular Weight247.27 g/mol g/mol
Typical Purity98.0-102.0% on dried basis (USP/EP); total impurities NMT 0.5%
Storage ConditionsStore in well-closed containers at 15-30 C, protected from light and moisture
Shelf Life60 months from date of manufacture
CategoryNitroimidazoles

Specifications are indicative and intended for sourcing reference only. Always confirm against the supplier's Certificate of Analysis and the applicable pharmacopeial monograph before issuing a purchase specification.

Typical Applications

Oral tablets for trichomoniasis, giardiasis, amoebiasis and bacterial vaginosis; fixed-dose combinations with ciprofloxacin, norfloxacin, ofloxacin, diloxanide furoate and fluconazole; IV infusion in some markets.

Manufacturers (1+)

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